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詳細(xì)介紹

朱功名,,男,博士,講師,,藥理學(xué)支部書記

聯(lián)系方式:[email protected]






教育經(jīng)歷:

20079-20116月??河南師范大學(xué)??生命科學(xué)學(xué)院

20119-20176月??蘭州大學(xué)????生命科學(xué)學(xué)院??碩博連讀??博士


工作經(jīng)歷:

20177-20187月??中山大學(xué)     特聘副研究員??藥物化學(xué)研究

20189-20235月??河南師范大學(xué)??化學(xué)化工學(xué)院

20235-至今???? 河南師范大學(xué)??抗病毒性傳染病創(chuàng)新藥物全國重點實驗室


研究領(lǐng)域與興趣:

1.核苷藥物設(shè)計合成及篩選

2.多肽藥物的定向合成及關(guān)鍵技術(shù)的開發(fā)

3.活性多肽后修飾及其化學(xué)生物學(xué)研究

4.核酸及多肽化學(xué)生物學(xué)研究


近年來主持的主要科研項目:

1.國家自然科學(xué)青年基金,,2019-2021年,,主持,,資助金額:27.5萬元,。

2.廣東省自然科學(xué)基金,,2018-2021年,,主持,資助金額:10萬元,。

3.博士后基金面上項目一等資助,,2018-2020年,主持,,資助金額:8萬元,。

4.河南師范大學(xué)博士啟動經(jīng)費,2019-2021年,,主持,,資助金額:8萬。

5.參與完成國家自然科學(xué)青年基金2項,,其中一項被評為優(yōu)秀,;

6.參與重點項目一項,面上項目兩項,。


代表性論文:

(1).Gongming Zhu#, Guangjun Bao#, Yiping Li, Wangsheng Sun,* Jing Li, Liang Hong,* and Rui Wang*. Efficient Catalytic Kinetic Resolution of Spiro-epoxyoxindoles with Concomitant Asymmetric Friedel-Crafts Alkylation of Indoles. Angew. Chem. Int. Ed. 2017, 56, 5332 –5335.

(2).Wangsheng Sun#, Gongming Zhu#, Chongyang Wu, Guofeng Li, Liang Hong,* and Rui Wang*. Organocatalytic Diastereo- and Enantioselective 1,3-Dipolar Cycloaddition of Azlactones and Methyleneindolinones. Angew. Chem. Int. Ed.2013, 52, 8633–8637.

(3).Gongming Zhu#, Yiping Li#, Guangjun Bao, Wangsheng Sun,* Liwu Huang, Liang Hong,* and Rui Wang*. Catalytic Kinetic Resolution of Spiro-Epoxyoxindoleswith 1 Naphthols: Switchable Asymmetric Tandem Dearomatization/Oxa-Michael Reaction and Friedel?Crafts Alkylation of 1 Naphthols at the C4 Position.ACS Catal.2018, 8, 1810?1816.

(4).Gongming Zhu, Guangjun Bao, Yiping Li, Junxian Yang, Wangsheng Sun, Jing Li, Liang Hong,* and Rui Wang*. Chiral Phosphoric Acid Catalyzed Asymmetric Oxidative Dearomatization of Naphthols with Quinones. Org. Lett., 2016, 18, 5288-5291.

(5).Gongming Zhu, Junxian Yang, Guangjun Bao, Ming Zhang, Jing Li, Yiping Li, Wangsheng Sun,* Liang Hong,* and Rui Wang*. Catalyst-controlled switch of regioselectivity in the asymmetric allylic alkylation of oxazolones with MBHCs,,Chem. Commun. 2016, 52, 7882-7885.

(6).Gongming Zhu, Wangsheng Sun, Chongyang Wu, Guofeng Li, Liang Hong,* and Rui Wang*. Base-Catalyzed Diastereoselective [3 + 3] Annulation of 3-Isothiocyanatooxindoles and Azomethine Imines. Org. Lett. 2013, 15, 4988.

(7).Jiaojiao Shen, Gongming Zhu, Yanbo You, Bianbian Huo, Fangyin Dai, Honglei Wang, Anlian Zhu and Lingjun Li. Designing a Light-Induced Glycosylation Reaction for Poststage Synthesis of ADP-2″-Deoxyribosyl Derivatives. Org. Lett. 2023, 21, 3961-3966.

(8).Mengqi Wang, Luyao Li, Shuping Yang, Fangyuan Guo, Gongming Zhu*, Bo Zhu*, Junbiao Chang*. Synthesis of novel oxazol-5-one derivatives containing chiral trifluoromethyl and isoxazole moieties as potent antitumor agents and the mechanism investigation. Bioorganic Chemistry. 2023, 135, 106505.

(9). Yuan-Yang Guo, Rujie Zhang, Bianbian Huo, Luying Wang, Donghe Yuan, Jingsi Bai, Honglei Wang, Gongming Zhu, Xiguang Zhang, Anlian Zhu, Tingjian Chen and Lingjun Li*. Site-specific unnatural base excision via visible light. Chem. Commun. 2022, 58, 11717-11720.

(10). Anlian Zhu; Xin Li; Lili Bai; Gongming Zhu; Yuanyang Guo; Jianwei Lin; Yiwen Cui; GaofeiTian; Lihe Zhang; Jianji Wang; Xiang David Li; Lingjun Li ; Biomimetic α-selective ribosylation enables two-step modular synthesis of biologically important ADP-ribosylated peptides, Nat. Commun., 2020, 11: 5600.