朱功名,,男,博士,講師,,藥理學(xué)支部書記
聯(lián)系方式:[email protected]
教育經(jīng)歷:
2007年9月-2011年6月??河南師范大學(xué)??生命科學(xué)學(xué)院
2011年9月-2017年6月??蘭州大學(xué)????生命科學(xué)學(xué)院??碩博連讀??博士
工作經(jīng)歷:
2017年7月-2018年7月??中山大學(xué) 特聘副研究員??藥物化學(xué)研究
2018年9月-2023年5月??河南師范大學(xué)??化學(xué)化工學(xué)院
2023年5月-至今???? 河南師范大學(xué)??抗病毒性傳染病創(chuàng)新藥物全國重點實驗室
研究領(lǐng)域與興趣:
1.核苷藥物設(shè)計合成及篩選
2.多肽藥物的定向合成及關(guān)鍵技術(shù)的開發(fā)
3.活性多肽后修飾及其化學(xué)生物學(xué)研究
4.核酸及多肽化學(xué)生物學(xué)研究
近年來主持的主要科研項目:
1.國家自然科學(xué)青年基金,,2019-2021年,,主持,,資助金額:27.5萬元,。
2.廣東省自然科學(xué)基金,,2018-2021年,,主持,資助金額:10萬元,。
3.博士后基金面上項目一等資助,,2018-2020年,主持,,資助金額:8萬元,。
4.河南師范大學(xué)博士啟動經(jīng)費,2019-2021年,,主持,,資助金額:8萬。
5.參與完成國家自然科學(xué)青年基金2項,,其中一項被評為優(yōu)秀,;
6.參與重點項目一項,面上項目兩項,。
代表性論文:
(1).Gongming Zhu#, Guangjun Bao#, Yiping Li, Wangsheng Sun,* Jing Li, Liang Hong,* and Rui Wang*. Efficient Catalytic Kinetic Resolution of Spiro-epoxyoxindoles with Concomitant Asymmetric Friedel-Crafts Alkylation of Indoles. Angew. Chem. Int. Ed. 2017, 56, 5332 –5335.
(2).Wangsheng Sun#, Gongming Zhu#, Chongyang Wu, Guofeng Li, Liang Hong,* and Rui Wang*. Organocatalytic Diastereo- and Enantioselective 1,3-Dipolar Cycloaddition of Azlactones and Methyleneindolinones. Angew. Chem. Int. Ed.2013, 52, 8633–8637.
(3).Gongming Zhu#, Yiping Li#, Guangjun Bao, Wangsheng Sun,* Liwu Huang, Liang Hong,* and Rui Wang*. Catalytic Kinetic Resolution of Spiro-Epoxyoxindoleswith 1 Naphthols: Switchable Asymmetric Tandem Dearomatization/Oxa-Michael Reaction and Friedel?Crafts Alkylation of 1 Naphthols at the C4 Position.ACS Catal.2018, 8, 1810?1816.
(4).Gongming Zhu, Guangjun Bao, Yiping Li, Junxian Yang, Wangsheng Sun, Jing Li, Liang Hong,* and Rui Wang*. Chiral Phosphoric Acid Catalyzed Asymmetric Oxidative Dearomatization of Naphthols with Quinones. Org. Lett., 2016, 18, 5288-5291.
(5).Gongming Zhu, Junxian Yang, Guangjun Bao, Ming Zhang, Jing Li, Yiping Li, Wangsheng Sun,* Liang Hong,* and Rui Wang*. Catalyst-controlled switch of regioselectivity in the asymmetric allylic alkylation of oxazolones with MBHCs,,Chem. Commun. 2016, 52, 7882-7885.
(6).Gongming Zhu, Wangsheng Sun, Chongyang Wu, Guofeng Li, Liang Hong,* and Rui Wang*. Base-Catalyzed Diastereoselective [3 + 3] Annulation of 3-Isothiocyanatooxindoles and Azomethine Imines. Org. Lett. 2013, 15, 4988.
(7).Jiaojiao Shen, Gongming Zhu, Yanbo You, Bianbian Huo, Fangyin Dai, Honglei Wang, Anlian Zhu and Lingjun Li. Designing a Light-Induced Glycosylation Reaction for Poststage Synthesis of ADP-2″-Deoxyribosyl Derivatives. Org. Lett. 2023, 21, 3961-3966.
(8).Mengqi Wang, Luyao Li, Shuping Yang, Fangyuan Guo, Gongming Zhu*, Bo Zhu*, Junbiao Chang*. Synthesis of novel oxazol-5-one derivatives containing chiral trifluoromethyl and isoxazole moieties as potent antitumor agents and the mechanism investigation. Bioorganic Chemistry. 2023, 135, 106505.
(9). Yuan-Yang Guo, Rujie Zhang, Bianbian Huo, Luying Wang, Donghe Yuan, Jingsi Bai, Honglei Wang, Gongming Zhu, Xiguang Zhang, Anlian Zhu, Tingjian Chen and Lingjun Li*. Site-specific unnatural base excision via visible light. Chem. Commun. 2022, 58, 11717-11720.
(10). Anlian Zhu; Xin Li; Lili Bai; Gongming Zhu; Yuanyang Guo; Jianwei Lin; Yiwen Cui; GaofeiTian; Lihe Zhang; Jianji Wang; Xiang David Li; Lingjun Li ; Biomimetic α-selective ribosylation enables two-step modular synthesis of biologically important ADP-ribosylated peptides, Nat. Commun., 2020, 11: 5600.