朱功名,男,博士,,副教授,綜合辦公室主任,,藥理學(xué)支部書記
聯(lián)系方式:[email protected]
教育經(jīng)歷:
2007年9月-2011年6月??河南師范大學(xué)??生命科學(xué)學(xué)院
2011年9月-2017年6月??蘭州大學(xué)????生命科學(xué)學(xué)院??碩博連讀??博士 導(dǎo)師:王銳院士
工作經(jīng)歷:
2017年7月-2018年7月??中山大學(xué) 特聘副研究員??藥物化學(xué)研究
2018年9月-2023年5月??河南師范大學(xué)??化學(xué)化工學(xué)院
2023年5月-至今???? 河南師范大學(xué)??抗病毒性傳染病創(chuàng)新藥物全國重點(diǎn)實(shí)驗(yàn)室
研究領(lǐng)域與興趣:
1.核苷藥物設(shè)計(jì)合成及篩選
2.多肽藥物的定向合成及關(guān)鍵技術(shù)的開發(fā)
3.活性多肽后修飾及其化學(xué)生物學(xué)研究
4.核酸及多肽化學(xué)生物學(xué)研究
近年來主持的主要科研項(xiàng)目:
1.國家自然科學(xué)青年基金,2019-2021年,,主持,,資助金額:27.5萬元。
2.廣東省自然科學(xué)基金,,2018-2021年,主持,,資助金額:10萬元,。
3.河南師范大學(xué)博士啟動(dòng)經(jīng)費(fèi),2019-2021年,,主持,,資助金額:8萬。
4.參與完成國家自然科學(xué)青年基金2項(xiàng),,其中一項(xiàng)被評(píng)為優(yōu)秀,;
5.參與國家重點(diǎn)研發(fā)計(jì)劃2項(xiàng),,重點(diǎn)項(xiàng)目1項(xiàng),面上項(xiàng)目3項(xiàng),。
獲得榮譽(yù):
2022年9月 獲評(píng)河南省優(yōu)秀學(xué)士論文指導(dǎo)教師,;
2023年6月 獲評(píng)河南師范大學(xué)“優(yōu)秀共產(chǎn)黨員”稱號(hào);
2023年12月 獲評(píng)河南師范大學(xué)“優(yōu)秀實(shí)習(xí)指導(dǎo)教師”,;
2024年6月 獲評(píng)河南師范大學(xué)“優(yōu)秀工會(huì)工作者”,。
代表性論文:
[1] Gongming Zhu#, Guangjun Bao#, Yiping Li, Wangsheng Sun,* Jing Li, Liang Hong,* and Rui Wang*. Efficient Catalytic Kinetic Resolution of Spiro-epoxyoxindoles with Concomitant Asymmetric Friedel-Crafts Alkylation of Indoles. Angew. Chem. Int. Ed. 2017, 56, 5332 –5335.
[2] Wangsheng Sun#, Gongming Zhu#, Chongyang Wu, Guofeng Li, Liang Hong,* and Rui Wang*. Organocatalytic Diastereo- and Enantioselective 1,3-Dipolar Cycloaddition of Azlactones and Methyleneindolinones. Angew. Chem. Int. Ed.2013, 52, 8633–8637.
[3] Gongming Zhu#, Yiping Li#, Guangjun Bao, Wangsheng Sun,* Liwu Huang, Liang Hong,* and Rui Wang*. Catalytic Kinetic Resolution of Spiro-Epoxyoxindoleswith 1 Naphthols: Switchable Asymmetric Tandem Dearomatization/Oxa-Michael Reaction and Friedel?Crafts Alkylation of 1 Naphthols at the C4 Position.ACS Catal.2018, 8, 1810?1816.
[4]Mengqi Wang, Shuping Yang, Xinge Li, Yingying Zheng, Yan Bai, Wenhan Luo, Gongming Zhu*, Junbiao Chang*, Bo Zhu*. Discovery of Novel Aromatic Urea-Imidazole Salt Derivatives for Cancer Therapy via Targeting ERK1/2, Journal of Medicinal Chemistry, 2025, 68, 4101-4132.
[5]Gongming Zhu,* Haiyang Zhang, Liyang Han, Honglei Wang, Anlian Zhu, Lingjun Li*. Solvent-Driven Room-Temperature Curtius Rearrangements to Access Nucleotides Bearing Substituted Fused Pyridones, Organic Letters, 2024, 26(20): 4356-4360.
[6] Gongming Zhu, Guangjun Bao, Yiping Li, Junxian Yang, Wangsheng Sun, Jing Li, Liang Hong,* and Rui Wang*. Chiral Phosphoric Acid Catalyzed Asymmetric Oxidative Dearomatization of Naphthols with Quinones. Org. Lett., 2016, 18, 5288-5291.
[7] Gongming Zhu, Junxian Yang, Guangjun Bao, Ming Zhang, Jing Li, Yiping Li, Wangsheng Sun,* Liang Hong,* and Rui Wang*. Catalyst-controlled switch of regioselectivity in the asymmetric allylic alkylation of oxazolones with MBHCs,Chem. Commun. 2016, 52, 7882-7885.
[8] Gongming Zhu, Wangsheng Sun, Chongyang Wu, Guofeng Li, Liang Hong,* and Rui Wang*. Base-Catalyzed Diastereoselective [3 + 3] Annulation of 3-Isothiocyanatooxindoles and Azomethine Imines. Org. Lett. 2013, 15, 4988.
[9] Jiaojiao Shen, Gongming Zhu, Yanbo You, Bianbian Huo, Fangyin Dai, Honglei Wang, Anlian Zhu and Lingjun Li. Designing a Light-Induced Glycosylation Reaction for Poststage Synthesis of ADP-2″-Deoxyribosyl Derivatives. Org. Lett. 2023, 21, 3961-3966.
[10]Mengqi Wang, Luyao Li, Shuping Yang, Fangyuan Guo, Gongming Zhu*, Bo Zhu*, Junbiao Chang*. Synthesis of novel oxazol-5-one derivatives containing chiral trifluoromethyl and isoxazole moieties as potent antitumor agents and the mechanism investigation. Bioorganic Chemistry. 2023, 135, 106505.