2. Erjun Hao, Dandan Fu, Dongchao Wang*, Tao Zhang, Guirong Qu,Gongxin Li,Yu Lan*, Haiming Guo*,Chemoselective Asymmetric Dearomative [3+2] Cycloaddition Reactions of Purines with Aminocyclopropanes,Org. Chem. Front. 2019,6,863-867. (SCI一區(qū),Top, IF=5.281)

3.Erjun Hao, Gong-Xin Li, Zhen-Zhen Lv, Fu-Sheng Li, Yu-Qing Chen, Shuang-Jie Lin, Cai-Zhe Shi, and Lei Shi*,“In-Situ Immobilization” of Multicomponent Chiral Catalyst (MCC) via Non-covalent Interactions for Heterogeneous Asymmetric Hydrogenation Reactions,Org. Chem. Front. 2020,7, 345-349. (SCI一區(qū),Top, IF=5.281)

4. Boyan Yu#, Erjun Hao#, Shaoming Fang#, Zhengqing Liu,Yongwei Wang, Zhenzhen Lv, Na Li, Xinyu Zhang, Lei Shi*, Yaping Du*,Controlled synthesis of high quality scandium-based nanocrystals as promising recyclable catalysts for silylcyanation reaction,Nanoscale,2017, 9(31), 10987-10991.(共同一作,SCI一區(qū), ,Top)
5. Peihua Zhao*, Kuankuan Xiong, Wenjun Liang, Erjun Hao*,Synthesis, crystal structures and electrocatalytic properties of bridgehead-C- functionalized diiron dithiolate complexes,J. Coord. Chem. 2015, 68,968-979.
6. Er-Jun Hao, Qing Zhang, Qi-ying Zhang*,Gui-Rong Qu, Xi-Ning Yang, Hai-Ming Guo*, Efficient Synthesis of Spirocyclic Nucleosides via Michael-initiated Intermolecular Cyclopropanation Reaction, Chin.J.Org.Chem. 2019, 39,3237-3243.
7. Erjun Hao, Xiaohan Jiang, Dandan Fu, Dongchao Wang*, Mingsheng Xie, Haiming Guo, Synthesis of 3-Cyanomethyl Oxoindoles via Palladium- catalyzed Domino Heck/Cyanation Reaction in Water, Chin.J.Org. Chem. 2016, 36, 2746-2751.
獲得榮譽(yù)與獎(jiǎng)勵(lì):
1、吉西他濱鹽酸鹽生產(chǎn)新工藝研究,河南省人民政府,河南省科技進(jìn)步三等獎(jiǎng)(證書(shū)編號(hào):2012-J-256-R05/06),2013;
2、河南師范大學(xué)優(yōu)秀教師;
3、河南師范大學(xué)優(yōu)秀班主任;
4、河南師范大學(xué)優(yōu)秀實(shí)習(xí)指導(dǎo)教師;
5、優(yōu)秀創(chuàng)新創(chuàng)業(yè)指導(dǎo)老師獎(jiǎng);
6、河南師范大學(xué)文明教師;
代表性授權(quán)發(fā)明專利:
1、[3+2]環(huán)加成不對(duì)稱脫芳構(gòu)化合成手性非芳香嘌呤核苷的方法,專利號(hào):ZL201810894271.4,第1發(fā)明人;
2、一種磷酸氟達(dá)拉濱的制備方法,專利號(hào):ZL201610278259.1,第1發(fā)明人;
3、一種合成2′-螺環(huán)基取代的三元碳環(huán)核苷的方法,專利號(hào):ZL201910374991.2,第1發(fā)明人。
English version:
Dr. Er-jun Hao
School of Chemistry and Chemical Engineering, Henan Normal University
Xinxiang, 453007, China
E-mail: [email protected]
Tel: +86-03733326335 or +86-15837307685.
Education and Academic career:
Lecturer, Henan Normal University, China(2008)
Ph.D.: Nankai University, China (2010, supervisor: Prof. Xiao-Qing Zhu and Prof. Jin-Pei Cheng)
M.S.: Henan Normal University, China (2005)
B.S.: Henan Normal University, China (2002)
Major Research Interests:
1. Design and synthesis of chiral nucleoside drugs;
2. Antitumor activity and structure-activity relationship study;
3. Photocatalytic asymmetric synthesis;
榮譽(yù)與獎(jiǎng)勵(lì):
1. “河南省科學(xué)技術(shù)進(jìn)步獎(jiǎng)三等獎(jiǎng)”(證書(shū)編號(hào):2012-J-256-R05/06),2013年;
2. 河南省科技廳科技成果鑒定:離子液體在藥物合成中的反應(yīng)介質(zhì)應(yīng)用研究,豫鑒字:第966號(hào),2012年;
3. 河南師范大學(xué)優(yōu)秀班主任;
4. 河南師范大學(xué)優(yōu)秀教師。
English version:Dr. Er-jun Hao
Henan Normal University
Xinxiang, 453007, China
E-mail: [email protected]
Tel:+86-03733326335 or +86-15837307685.
Education and Academic career:
Lecturer, Henan Normal University, China(2008)
Ph.D.: Nankai University, China (2010, supervisor: Prof. Xiao-Qing Zhu and Prof. Jin-Pei Cheng)
M.S.: Henan Normal University, China (2005,supervisor: Prof. Wei Li)
B.S.: Henan Normal University, China (2002,supervisor: Prof. Yu-Lu Wang )
Major Research Interests:
1. Design and synthesis of chiral nucleoside drugs;
2. Antitumor activity and structure-activity relationship study;
3. Photocatalytic asymmetric synthesis;